Table 1.
Zap‐Pano shows little KDAC inhibition in vitro.
IC50 values (nM) for Pano and Zap‐Pano against KDAC1‐9 and KDAC11. The colour scale represents a heat map, with ‘hot’ colours showing effective enzyme inhibition. [a] Data obtained by Reaction Biology Corporation, NI=no inhibition observed at concentrations up to 10 μM. [b] Data taken from Arts et al. [39]