Table 2.
Compounds on inhibitory activities of PI3Ks.
| Compounds | IC50 (μM)∗ | |||
|---|---|---|---|---|
| PI3Kα | PI3Kβ | PI3Kγ | PI3Kδ | |
| TAN | >40 | >40 | 17.72 ± 1.16 | >40 |
| LUT | 2.49 ± 0.34 | 2.95 ± 0.19 | 5.79 ± 0.10 | 1.55 ± 0.15 |
| HES | >40 | >40 | >40 | >40 |
| NAR | >40 | >40 | >40 | >40 |
| AUR | >40 | >40 | 13.75 ± 1.31 | >40 |
| PI103 (nM) | 7.10 ± 0.14 | 13.50 ± 0.60 | 85.50 ± 1.88 | 12.50 ± 2.07 |
∗ Values are means of three independent experiments.