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. 2022 Jul 13;2022:2156157. doi: 10.1155/2022/2156157

Table 2.

Compounds on inhibitory activities of PI3Ks.

Compounds IC50 (μM)
PI3Kα PI3Kβ PI3Kγ PI3Kδ
TAN >40 >40 17.72 ± 1.16 >40
LUT 2.49 ± 0.34 2.95 ± 0.19 5.79 ± 0.10 1.55 ± 0.15
HES >40 >40 >40 >40
NAR >40 >40 >40 >40
AUR >40 >40 13.75 ± 1.31 >40
PI103 (nM) 7.10 ± 0.14 13.50 ± 0.60 85.50 ± 1.88 12.50 ± 2.07

Values are means of three independent experiments.