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In‐vitro (FRET) and in‐cellulo (BRET) binding data of selected inhibitors.
|
Compound |
FRET assay (IC50) [nM] |
BRET assay (EC50) [nM] |
|---|---|---|
|
vorinostat (6) |
200[a] |
630[a] |
|
quisinostat (11) |
10 |
40[a] |
|
abexinostat (12) |
4 |
8[a] |
|
tubastatin A (14) |
19 |
13[a] |
|
48 a |
5 |
26 |
|
48 b |
2 |
10 |
[a] From Géraldy et al. [32]
