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Table 2.
In vitro inhibitory activity of hybrids 9g and 9k towards EGFR.
| |
|---|---|
| Compound | IC50 (nM) |
| EGFR | |
| 9g | 267 ± 12 |
| 9k | 395 ± 17 |
| Erlotinib | 57 ± 3 |