Table III.
Composition and Characterization of Prepared Solid Dispersion
| Compositions | Characterization | ||||||
|---|---|---|---|---|---|---|---|
| Polymer | Formulation code | Drug carrier ratio | % yield | % drug content | Particle size | Solubility mg/ml | PDI |
| BEX | - | - | - | - | 0.00018 | - | |
| BEX-POLO1 | 1:1 | 92.5±0.8 | 96.1±1.3 | 825.0±7.1 | 0.00162 | 0.302±21.3 | |
| BEX-POLO2 | 1:2 | 85.2±1.2 | 96.9±1.4 | 721.8±9.1 | 0.00206 | 0.401±18.9 | |
| POLO | BEX-POLO3 | 1:3 | 82.9±1.1 | 97.5±1.1 | 694.1±3.5 | 0.00272 | 0.376±11.1 |
| BEX-POLO4 | 1:4 | 79.5±0.9 | 98.4±1.0 | 515.2±4.2 | 0.00356 | 0.448±14.1 | |
| BEX-POLO5 | 1:5 | 73.6±1.0 | 99.1±1.1 | 471.5±5.3 | 0.00361 | 0.396±10.8 | |
| BEX-MLBG1 | 1:1 | 94.7±0.8 | 96.3±1.8 | 918.3±7.1 | 0.00153 | 0.089±8.8 | |
| BEX-MLBG2 | 1:2 | 95.0±1.1 | 97.1±1.1 | 875.9±6.5 | 0.00211 | 0.115±11.0 | |
| MLBG | BEX-MLBG3 | 1:3 | 94.1±1.2 | 96.8±1.4 | 795.3±7,1 | 0.00284 | 0.101±10.9 |
| BEX-MLBG4 | 1:4 | 95.1±1.4 | 99.0±1.2 | 745.7±4.4 | 0.00340 | 0.042±15.9 | |
| BEX-MLBG5 | 1:5 | 95.4±0.9 | 97.1±1.7 | 605.8±5.3 | 0.00344 | 0.095±11.8 | |