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. 2022 Jul 18;24(29):5376–5380. doi: 10.1021/acs.orglett.2c02050

Table 1. Influence of Lewis Basicity on N–F Bond Activation of Selectfluora.

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a

Reaction conditions: 4-fluorophenylacetlc acid (0.3 mmol), Selectfluor (0.36 mmol), DMAP (0.6 mmol), MeCN (1.5 mL), rt, 4 h.

b

Converaion of 4-fluorophenylacetic acid determined by 1H NMR using dimethyl maleate as an internal standard.

c

NMR yield determined by 1H NMR using dimethyl maleate as an internal standard.