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. 2022 Jul 22;18:889–915. doi: 10.3762/bjoc.18.90

Scheme 3.

Scheme 3

Synthesis of 2-aryl-1-methyl-2,3-dihydrobenzo[c][1,2]azaphosphole 1-oxides 13 from N-aryl-2-chloromethylphenyl(methyl)phosphinamides 12.