Table 2. Reduction of Pentylenetetrazol (70 mg/kg) Produced Lethality by KRM-II-81 and Its HCl Salt.
compound | lethality/number tested | latency to death (s) |
---|---|---|
vehicle | 4/7 | 25.75 ± 8.02 |
KRM-II-81 (2 h) | 0/6a | |
KRM-II-81 (4 h) | 0/6a | |
KRM-II-81 (8 h) | 0/6a | |
KRM-II-81·HCl (2 h) | 0/6a | |
KRM-II-81·HCl (4 h) | 1/6 | 15.68 |
KRM-II-81·HCl (8 h) | 1/6 | 43.00 |
P < 0.05.