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. 2022 Jul 27;7(31):27550–27559. doi: 10.1021/acsomega.2c03029

Table 2. Reduction of Pentylenetetrazol (70 mg/kg) Produced Lethality by KRM-II-81 and Its HCl Salt.

compound lethality/number tested latency to death (s)
vehicle 4/7 25.75 ± 8.02
KRM-II-81 (2 h) 0/6a  
KRM-II-81 (4 h) 0/6a  
KRM-II-81 (8 h) 0/6a  
KRM-II-81·HCl (2 h) 0/6a  
KRM-II-81·HCl (4 h) 1/6 15.68
KRM-II-81·HCl (8 h) 1/6 43.00
a

P < 0.05.