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. 2022 Jul;10(14):806. doi: 10.21037/atm-22-3136

Table 2. Summary of the mechanism of hesperetin in the treatment of cerebral ischemia.

Effect Mechanism References
Anti-oxidative stress and apoptosis Inhibit ROS, LPO, and JNK/Bax, caspase-3 (46-50)
Promote Nrf2, HO-1, and Bcl-2
Anti-atherosclerosis Inhibit TNF-α, MCP-1, and the G0/G1 phase (56)
Promote adenosine triphosphate binding transporter A1
Anti-inflammatory reaction Inhibit P-NF-κB, ERK1/2, and p38 MAPK (58-60)
Anti-thrombosis Inhibit PCL-2, phosphorylation, and cyclooxygenase-1 (24)
Anti-hyperlipidemia Inhibit HMG-CoA reductase and ACAT enzymes (65)
Assembled lipid for carrier protein binding
Transcription of ACAT-2 mRNA
Anti-nitric oxide damage Inhibit iNOS (66,68)

ROS, reactive oxygen species; LPO, lipid peroxidation; JNK, c-Jun N-terminal kinase; BAX, Bcl-2 associated X protein; Nrf-2, nuclear factor erythroid 2-related factor 2; HO-1, heme oxygenase-1; Bcl-2, B cell lymphoma-2; TNF-α, tumor necrosis factor-α; MCP-1, monocyte chemoattractant protein-1; p-NF-κB, phosphorylated -nuclear factor-kappaB; ERK1/2, extracellular signal-regulated kinase 1/2; p38 MAPK, p38 mitogen-activated protein kinase; PLC-2, phospholipase C-2; HMG CoA, 3-hydroxy-3-methylglutaryl-coenzyme A; ACAT, acyl coenzyme cholesterol acyltransferase; iNOS, inducible nitric oxide synthase.