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. 2022 Aug 8;8(8):e10101. doi: 10.1016/j.heliyon.2022.e10101

Table 15.

Drug likeness assessment of the lead compounds based on Ghose, Veber, Egan, Muegge, QED, and Synthetic accessibility scores.

Molecule Ghose Veber Egan Muegge QED SA score
9 Yes No No No 0.62 3.148
10 Yes No No No 0.582 3.215
11 Yes No No No 0.582 3.158
17 Yes No No No 0.549 3.25
22 Yes No No No 0.515 3.32
31 Yes No No No 0.554 3.272
Oseltamivir Yes Yes Yes Yes 0.213 4.392
Zanamivir Yes Yes Yes Yes 0.691 3.758

Key: Quantitative Estimate of Drug-likeness (QED), Synthetic accessibility (SA) score.