TABLE 5.
Pharmacokinetic parameters of rivaroxaban per p.o. administration.
Parameter | Rivaroxaban | Rivaroxaban + imatinib | Rivaroxaban + gefitinib | Rivaroxaban + sunitinib |
---|---|---|---|---|
AUC(0-t) | 1.547 ± 0.268 | 2.946 ± 0.647 * | 1.587 ± 0.145 | 0.583 ± 0.101 ** |
Cmax | 129.7 ± 22.70 | 281.4 ± 54.05 ** | 106.8 ± 23.60 | 35.60 ± 2.426 ** |
Tmax | 4 | 3 | 3 | 4 |
AUC(0-t) was recorded as ug/mL·h, Cmax was recorded as ng/mL, and Tmax was recorded as h. Data are expressed as the mean ± S.D.
p < 0.05.
p < 0.01 compared with control; n = 5.