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. 2022 Aug 22;13:914842. doi: 10.3389/fphar.2022.914842

TABLE 7.

Comparison of ChemScore values of TKIs binding to CYP2J2, CYP3A4, BCRP, and P-gp.

TKIs CYP2J2 CYP3A4 BCRP P-gp
Imatinib −30.296 −49.611 −31.524 −29.995
Gefitinib −33.232 −38.264 −30.913 −29.384
Sunitinib −25.039 −38.026 −28.127 −25.905