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. 2022 Aug 24;14(17):4094. doi: 10.3390/cancers14174094

Table 2.

Treatment responses in individual patients.

Samples Hit Compounds
Sample 1 (+)-JQ1, (S)-HDAC-42 (AR-42), 2′-Deoxy-5-fluorocytidine, 5-Iodotubercidin, ACY-1215 (Rocilinostat), Apicidin, BI-2536, BML-281, Bromosporine, CAY10603, CBHA, Chidamide, CPI203, CUDC-101, CUDC-907 (Fimepinostat), Disulfiram, Entinostat (MS-275), Fluoro-SAHA, Givinostat (ITF2357), I-BET 151, I-BET62 (GSK525762), JIB 04, JNJ-26481585, KD 5170, LAQ824 (Dacinostat), LMK 235, LSD1-C12, M-344, NSC-3852, Oxamflatin, PXD101 (Belinostat), Pyroxamide, SAHA, SB 939 (Pracinostat), Scriptaid, Suberoyl bis-hydroxamic acid, TG101348 (SAR302503), Trapoxin A, Trichostatin A, β-Lapachone
Sample 2 (+)-JQ1, (S)-HDAC-42 (AR-42), 5-Iodotubercidin, Apicidin, BI-2536, CBHA, CPI203, CUDC-907 (Fimepinostat), Entinostat (MS-275), Fluoro-SAHA, Givinostat (ITF2357), I-BET 151, I-BET62 (GSK525762), JNJ-26481585, LAQ824 (Dacinostat), LMK 235, M-344, Nexturastat A, NSC-3852, Oxamflatin, PCI-24781 (Abexinostat), PXD101 (Belinostat), SAHA, SB 939 (Pracinostat), Scriptaid, Trapoxin A, Trichostatin A, β-Lapachone
Sample 3 (S)-HDAC-42 (AR-42), CUDC-907 (Fimepinostat), Disulfiram, Entinostat (MS-275), Givinostat (ITF2357), JIB 04, JNJ-26481585, LAQ824 (Dacinostat), LMK 235, M-344, NSC-3852, Oxamflatin, PCI-24781 (Abexinostat), PXD101 (Belinostat), SAHA, SB 939 (Pracinostat), Trapoxin A, Trichostatin A
Sample 4 (+)-JQ1, (S)-HDAC-42 (AR-42), 5-Iodotubercidin, ACY-1215 (Rocilinostat), Apicidin, BI-2536, Bromosporine, CBHA, Chidamide, CI-994, CPI203, CUDC-101, CUDC-907 (Fimepinostat), Disulfiram, DZNep, Entinostat (MS-275), EP-336, Fluoro-SAHA, Givinostat (ITF2357), I-BET 151, I-BET62 (GSK525762), JIB 04, JNJ-26481585, LAQ824 (Dacinostat), LMK 235, M-344, Nexturastat A, NSC-3852, Oxamflatin, PCI-24781 (Abexinostat), PXD101 (Belinostat), SAHA, SB 939 (Pracinostat), Scriptaid, TG101348 (SAR302503), Trapoxin A, Trichostatin A, β-Lapachone
Sample 5 (+)-JQ1, (S)-HDAC-42 (AR-42), BI-2536, CPI203, CUDC-907 (Fimepinostat), Disulfiram, Entinostat (MS-275), Givinostat (ITF2357), I-BET62 (GSK525762), JNJ-26481585, LAQ824 (Dacinostat), LMK 235, NSC-3852, Oxamflatin, PXD101 (Belinostat), SB 939 (Pracinostat), Trapoxin A, Trichostatin A
Sample 6 (+)-JQ1, (S)-HDAC-42 (AR-42), 5-Iodotubercidin, Apicidin, BI-2536, CPI203, CUDC-907, Disulfiram, Entinostat (MS-275), EP670, Fluoro-SAHA, Givinostat (ITF2357), -BET 151, I-BET62 (GSK525762), JIB 04, JNJ-26481585, LAQ824 (Dacinostat), LMK 235, M-344, NSC-3852, Oxamflatin, PXD101 (Belinostat), SB 939 (Pracinostat), Scriptaid, Trapoxin A, Trichostatin A
Sample 7 (+)-JQ1, (S)-HDAC-42 (AR-42), Apicidin, BI-2536, CPI203, CUDC-907, Entinostat (MS-275), JNJ-26481585, LAQ824 (Dacinostat), LMK 235, M-344, NSC-3852, Oxamflatin, PXD101 (Belinostat), Trapoxin A, Trichostatin A
Sample 8 (+)-JQ1, (S)-HDAC-42 (AR-42), 5-Iodotubercidin, Apicidin, CBHA, CPI203, CUDC-907, Entinostat (MS-275), EP670, Givinostat (ITF2357), JNJ-26481585, LAQ824, LMK235, M-344, Nexturastat A, NSC-3852, OLAPAR 1B, Oxamflatin, PXD101 (Belinostat), SB 939 (Pracinostat), Scriptaid, Trapoxin A, Trichostatin A
Sample 9 (+)-JQ1, (S)-HDAC-42 (AR-42), 2′-Deoxy-5-fluorocytidine, 5-Iodotubercidin, AK-7, Apicidin, BI-2536, BML-266, CBHA, CI-994, CPI203, CTPB, CUDC-907, Disulfiram, DZNep, Entinostat (MS-275), EP670, EPZ-5676, Fluoro-SAHA, Givinostat (ITF2357), GSK126, GSK-J1, I-BET 151, I-BET762 (GSK525762), JIB 04, JNJ-26481585, LAQ824, LMK 235, LSD1-C12, LY294002, M-344, MM-102, Nexturastat A, Nicotinamide, NSC-3852, OG-L002, OLAPAR 1B, Oxamflatin, P22077, PBIT, PTC-209, Piceatannol, PXD101 (Belinostat), Pyroxamide, RG 108, RGFP966, RN-1, SAHA, SB 939 (Pracinostat), SBHA, SBI-7673, Scriptaid, SGI-1027, TC-H 106, TCS HDAC6 20b, TG101348 (SAR302503), Trapoxin A, Trichostatin A