. 2022 Aug 3;13(9):1434–1443. doi: 10.1021/acsmedchemlett.2c00173

Table 3. Compounds Screened in the Fragment-Growing Campaign^a.

n.d. = not determined: *Residual activity >50% when tested in single dose at 100 μM. ^#Compound rapidly crystallizing in the protein and assay buffers.

Table 3. Compounds Screened in the Fragment-Growing Campaigna.

Table 3. Compounds Screened in the Fragment-Growing Campaign^a.