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. 2022 Sep 12;15:132. doi: 10.1186/s13045-022-01320-5

Table 3.

pH-responsive building blocks for tumor treatment

pH-sensitive building block Therapeutic agent Tumor model Therapeutic application Refs.
Poly(2-(hexamethyleneimino)ethyl methacrylate siBRD4-loaded TCPA2-NPs Prostatic cancer LNCaP-bearing mouse GT [477]
HRNMs Glioblastoma Chemotherapy [478]
Poly(diisopropanol amino ethyl methacrylate) GPDPA NPs Glioblastoma Chemotherapy PTT [479]
Benzoic-imine bond CA-MTX NPs Cervical carcinoma Chemotherapy [480]
nBSA-Dox Hepatocellular carcinoma Chemotherapy [481]
NdIIIIP-N = CH-PEG Cervical carcinoma Chemotherapy PTT [482]
DOX-ICM Glioblastoma Chemotherapy [483]
Au@PP/RA/siRNA Pancreatic cancer Chemotherapy [484]
Pyridine-2-imine Gold nanomachine Breast cancer PTT [485]
PMNP-DOX@RBC Breast cancer Chemotherapy, CDT [486]
Amide bond DOX-CC-NP Squamous cell carcinoma Chemotherapy [19]
PDNBF NPs Breast cancer Chemotherapy PTT [487]
Nanodrug complex MONCs Breast cancer Chemotherapy PDT [488]
B780/Qu NPs Breast cancer Chemotherapy PDT, PTT [98]
Gadolinium oxide Gd2O3 NSs Melanoma Chemotherapy [489]
FS-GdNDs Breast cancer PTT [490]
Triplex DNA sequence NLNs/DOX Breast cancer Chemotherapy [491]
DNA Conjugated AuNPs Breast cancer Chemotherapy PTT [492]