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. 2011 Jun;20(120):71–84. doi: 10.1183/09059180.00000511

Table 2. Pharmacological management of multi-drug resistant (MDR) tuberculosis (TB).

First-line oral drugs Injectable bactericidal drugs# Fluoroquinolones# Second-line bacteriostatic drugs Other drugs with unclear or unproven efficacy
Rifampicin Streptomycin Moxifloxacin Cycloserine Clofazimine
Isoniazid Amikacin Gatifloxacin p-aminosalicyclic acid Clarithromycin
Rifabutin Kanamycin Ofloxacin Prothionamide Amoxicillin/clavulanate
Ethanmbutol Capreomycin Levofloxacin Ethionamide Linezolid
Pyrizinamide Terizidone Imipenem/cilastatin
Thioacetazone
High-dose isoniazid
Order in which drugs are added to MDR-TB regimen →

#: all MDR-TB regimens should include one injectable and one fluoroquinolone where possible; : by definition, isolates classed as MDR will be resistant to these drugs.