| AB3 | Anti-cancer drug |
| ABDA | 9,10-Anthracenediyl-bis(methylene) dimalonic acid |
| ABMDMA | 9,10-Anthracenediyl-bis(methylene)dimalonic acid |
| ABS | Acetate buffer solution |
| ADPA | 10-dipropionic acid, disodium salt |
| AEP | 2-aminoethyl dihydrogen phosphate |
| AFM | Atomic force microscope |
| ATF | Amino terminal fragment of urokinase plasminogen activator |
| AuNPs | Gold nanoparticles |
| Azo | Azobenzene |
| BFNS | Bifunctional nanospheres |
| BP | Bis-pyrene |
| bPEI | Branched polyethylenimine |
| BRET | Bioluminescence resonance energy transfer |
| BSA | Bovine serum albumin |
| BTSA | Bis(trimethylsilyl)acetamide |
| BT | Barium–titanate |
| CaB | Cathepsin B |
| CD | Cyclodextrin |
| cDDP | Cis-diaminedichloroplatine(II) |
| Ce6 | Chlorin e6 |
| CLSM | Confocal laser scanning microscopy |
| CQDs | Carbon quantum dots |
| CR | Core–satellite superstructure |
| C18RB | Hydrocarbonized RB |
| Cs-Na | Nitroimidazole-modified chitosan |
| CTAB | Cetyltrimethylammoniumbromide |
| CTS | Chitosan |
| Cy3 | Cyanine 3 |
| DCFH-DA | Dichlorodihydrofluorescein-diacetate |
| DLS | Dynamic light scattering |
| DMA | 9,10-Dimethylanthracene |
| DNA | Deoxyribonucleic acid |
| DOX | Doxorubicin |
| DPBF | 1,3-diphenylisobenzofuran |
| EADC | 1-Ethyl-3-(3-dimethylaminopropyl)carbodiimide |
| EDC | N-Ethyl-N′-(3-(dimethylamino)propyl)carbodiimide |
| EPR | Enhanced permeability effect |
| FA | Folic acid |
| FITS | Fluorescein isothiocyanate |
| FRET | Förster resonance energy transfer |
| 5FU | 5-Fluorouracil |
| GG | Guar gum |
| GRDs | Gadolinium-rose bengal coordination polymer nanodots |
| GSH | Glutathione |
| HA | Hyaluronic acid |
| HAx | Hexamethylenediamine |
| HCPT | 10-Hydroxycamptothecin |
| HMSNs | Hollow mesoporous silica nanoparticles |
| HSPC | Hydrogenated soy L-a-phosphatidylcholine |
| IR | Infrared |
| IR825 | NIR-absorbing dye |
| LIFU | Low-intensity focused ultrasound |
| Ln | Lanthanide |
| LNP | Luminescent lanthanide nanoparticles |
| MB | Methylene blue |
| MF | Multifunctional |
| MMSN | Magnetic mesoporous silica nanoparticle |
| MNCs | Magnetic nanoclusters |
| Mo | Oxymolybdate |
| MOF | Metal–organic frameworks |
| MRI | Magnetic resonance imaging |
| MS | Mesoporous silica |
| MSNs | Mesoporous silica nanoparticles |
| MTD | Maximum tolerated dose |
| MTT | 3-[4,5-Dimethylthiazol-2-yl]-2,5 diphenyl tetrazolium bromide |
| MUCNPs | Multi-shelled upconversion nanoparticles |
| NCs | Nanocarriers |
| Nd | Not determined |
| NHS | N-Hydroxysuccinimide |
| NIR | Near infrared |
| NPs | Nanoparticles |
| OA | Oleic acid |
| 1O2 | Singlet oxygen |
| PAA | Polyacrylic acid |
| PAH | Poly(allylamine) |
| PAMAM | Poly(amidoamine) |
| PARN | Amphiphilic peptide nanocapsules |
| PBS | Phosphate buffer solution |
| PCL | PEG-block-poly(ε-caprolactone) |
| Pdots | Polymer dots |
| PDT | Photodynamic therapy |
| PE | Phosphoethanolamine |
| PEG | Polyethyleneglycol |
| PEG-b-PAsp | Polyethylene glycol-b-poly(aspartic acid) |
| PEI | Polyethylene imine |
| PE-NH2 | 1,2-Dioleoyl-sn-glycero-phosphoethanolamine-N(hexanoylamine) |
| PFH | Perfluorohexane |
| PGA | Poly(glycolic acid) |
| PHLA | Partially hydrolyzed α-lactalbumin |
| p.i | Post injection |
| PLA | Poly(lactic acid) |
| PLGA | Poly(lactic-co-glycolic acid) |
| PPADT | Poly-(1,4-phenyleneacetone dimethylenethioketal) |
| PS | Photosensitizer |
| PTT | Photothermal therapy |
| PTX | Paclitaxel |
| PVA | Poly(vinyl alcohol) |
| PVK | Poly(N-vinyl carbazole) |
| QDs | Quantum dots |
| QSY7 | ROS quenching |
| RB | Rose Bengal |
| RBD | Rose bengal ω-carboxyheptyl ester |
| RET | Resonance energy transfer |
| ROS | Reactive oxygen species |
| ScNPs | Scintillating nanoparticles |
| SHG | Second harmonic generation |
| SOSG | Singlet oxygen sensor green |
| SSTRs | Somatostatin receptors |
| TEM | Transmission emission microscopy |
| TEOS | Tetraethyl orthosilicate |
| TMP–OH | 2,2,6,6-Tetramethyl-4-piperidinol |
| TOPO | Trioctylphosphine oxide |
| TPA | Two-photon activation |
| TUNEL | Terminal deoxynucleotidyl transferase dUTP nick end labeling |
| UCL | Upconversion luminescence |
| UCNPs | Upconversion nanoparticles |
| UPA | Urokinase plasminogen activator |
| US | Ultrasound |
| UV | Ultraviolet |
| WEN | White emitting NaYF4 |
| XLNPs | X-ray-luminescent nanoparticles |
| X-PDT | Photodynamic therapy induced by X-ray |
| ZIF-90 | Zeolitic imidazolate framework-90 |
| ZnPc-COOH | Zinc β-carboxyphthalocyanine |