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. 2022 Aug 25;15(9):1050. doi: 10.3390/ph15091050

Table 4.

IC50 values of compounds 4h, 4j, 4k, and 4q against DAPK1 kinase.

Cpd DAPK1 a, IC50 (μM)
4h 6.81
4j 1.70
4k 7.26
4q 1.09

a Mean values of duplicate mode 10-dose IC50 assays with DAPK1 kinase, with 3-fold serial dilution starting at 10 μM.