Table 4.
IC50 values of compounds 4h, 4j, 4k, and 4q against DAPK1 kinase.
| Cpd | DAPK1 a, IC50 (μM) |
|---|---|
| 4h | 6.81 |
| 4j | 1.70 |
| 4k | 7.26 |
| 4q | 1.09 |
a Mean values of duplicate mode 10-dose IC50 assays with DAPK1 kinase, with 3-fold serial dilution starting at 10 μM.
IC50 values of compounds 4h, 4j, 4k, and 4q against DAPK1 kinase.
| Cpd | DAPK1 a, IC50 (μM) |
|---|---|
| 4h | 6.81 |
| 4j | 1.70 |
| 4k | 7.26 |
| 4q | 1.09 |
a Mean values of duplicate mode 10-dose IC50 assays with DAPK1 kinase, with 3-fold serial dilution starting at 10 μM.