Skip to main content
. 2022 Sep 23;42(9):BSR20221789. doi: 10.1042/BSR20221789

Table 1. Multifunctional AMP in clinical trials.

Peptide name Administration Phase Target Structure
Gramicidin Topical III Infected wounds and ulcers Polycyclic lantibiotic
Polymixin B Topical III Gram-negative bacteria Cyclic polypeptide
Polymixin E (Colistin) Intravenus III A. baumannii/Pneumonia Cyclic polypeptide
Daptomycin Intravenous III Skin infection/bacteremia Lipopeptide
LL-37 Topical II Leg ulcers Human cathelicidn
Melittin Intradermal I/II Inflammation Alpha-helical peptide
Pexiganan (MSI-78) Topical III Diabetic foot ulcers Alpha-helical peptide
Omiganan (MBI-226) Topical III Antisepsis/catheter infections Derivative of indolicidine
OP-145 Ear drops I/II Chronic middle ear infection Derivative of LL-37
P113 (PAC-113) Mouth rinse II Oral candidiasis Fragment of histatin-5
hLF1-11 Intravenous I/II Bacterial/fungal infections Fragment of human lactoferrin
DPK-060 Ear drops II Acute external otitis Derivative of kininogen
AP-214 Intravenous II Postsurgical organ failure Derivative of α-MSH
PMX-30063 Intravenous II Acute bacterial skin infection Defensin mimetic