Skip to main content
. 2022 Sep 12;13:947252. doi: 10.3389/fphar.2022.947252

TABLE 1.

Scores and mechanisms of 20 potential drugs.

Name Comprehensive Score MOA (mechanism of action)
AS-703026 98.41 MEK inhibitor
ISOX 96.26 HDAC inhibitor
apicidin 96.09 HDAC inhibitor
MST-312 96.02 telomerase inhibitor
WT-171 94.31 HDAC inhibitor
cytochalasin-b 94.27 microtubule inhibitor, phagocytosis inhibitor
vorinostat 92.59 HDAC inhibitor, cell cycle inhibitor
epoxycholesterol 91.54 LXR agonist
WYE-354 91.21 mTOR inhibitor
SB-590885 91.06 RAF inhibitor
cytochalasin-d 89.01 Actin polymerization inhibitor, actin stabilizer
THM-I-94 88.99 HDAC inhibitor, apoptosis stimulant, cell cycle inhibitor
WYE-125132 88.82 mTOR inhibitor, PI3K inhibitor
trichostatin-a 87.17 HDAC inhibitor, CDK expression enhancer, ID1 expression inhibitor
wortmannin 86.89 PI3K inhibitor, ATM kinase inhibitor, PLK inhibitor, etc.
torin-2 86.04 mTOR inhibitor
BI-2536 85.47 PLK inhibitor, apoptosis stimulant, cell cycle inhibitor, protein kinase inhibitor
fluticasone 85.25 Glucocorticoid receptor agonist
WAY-170523 85.1 Metalloproteinase inhibitor
fenpiverinium 85.05 Acetylcholine receptor antagonist