| Nomenclature | Estrogen receptor‐α | Estrogen receptor‐β |
| Systematic nomenclature | NR3A1 | NR3A2 |
| HGNC, UniProt | ESR1 , P03372 | ESR2 , Q92731 |
| Endogenous agonists | estriol [73], estrone [73] | – |
| Selective agonists | propylpyrazoletriol [72, 133], ethinylestradiol [61] | WAY200070 [91], diarylpropionitrile [98, 133], prinaberel [27, 91] |
| Sub/family‐selective antagonists | bazedoxifene (pIC50 7.6) [101] | bazedoxifene (pIC50 7.1) [101] |
| Selective antagonists | clomiphene (pKi 8.9) [3], methyl‐piperidino‐pyrazole (pKi 8.6) [137] | R,R‐THC (pKi 8.4) [97, 138], PHTPP (pKi 6.9) [168] |
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