(A) Primary hippocampal cultures were treated on day
in vitro 2 (DIV2) with sonicated, preformed
α-synuclein fibrils (1 μg/mL) and immunostained on DIV12 for
somatodendritic neuron marker MAP2, neuronal process marker β-tubulin
III, APE1, and phosphorylated α-synuclein (pSer129; also
see
Fig. S1-S2). Nuclei were stained with the
Hoechst reagent. (B-E) Primary hippocampal cultures were treated on
DIV2 with α-synuclein fibrils (1 μg/mL) and APE1-targeted shRNA by
lentiviral delivery (60,000 transduction units per well in 96-well plates).
Cells were fixed three days (B) or 10 days (C-E) after
lentiviral exposure and stained for pan-nuclear markers DRAQ5 or Hoechst
(also see
Fig. S3-S5). (B) APE1 levels
are shown as a fraction of DRAQ5+ nuclear staining on DIV5 via
In-Cell Western analyses on a 16-bit, low resolution/high sensitivity infrared
imager. (C-E) Microscopic quantification of DRAQ5+ cell
counts, pSer129+ inclusion sizes (fold-change of nontargeting
controls), and pSer129+ inclusion densities on DIV12 after APE1
knockdown. (F-J) Primary hippocampal cultures were treated on DIV2
with α-synuclein fibrils (1 μg/mL) and APE1 Inhibitor III. Cells
were immunostained on DIV12 for pSer129 and APE1 (see
Fig. S6).
(F) Hoechst+ cell counts and (G)
APE1+ cell counts as % of untreated controls. (H)
pSer129+ inclusion size (fold-change of untreated controls).
(I) pSer129+ inclusion counts as a fraction of
Hoechst+ cell numbers (fold-change of untreated controls).
(J) Subcellular localization of the inclusions was not changed
by APE1 inhibitor III treatment (Fig. S1D
for higher-resolution images and reference to white arrow).
Data are shown as mean ± S.D. of 3-4 independent cultures. For
B-I, two-way ANOVAs were followed by the Bonferroni
post hoc (except D and H, which
were analyzed with one-way ANOVA/Bonferroni). For B-E,
*p≤0.05, **p≤0.01 shRNA vs.
non-targeting lentivirus control; +++p≤0.001 vehicle vs.
fibrils. For F-I, *p≤0.05,
**p≤0.01 APE1 inhibitor III vs. untreated (UT) or
DMSO controls; +++p≤0.001 vehicle vs. fibrils.