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. 2022 Sep 28;13:95. doi: 10.1007/s12672-022-00559-1

Table 2.

Characteristics of included study

Author, year Registered number,
Acronym
Phase Region Study design Baseline characteristics of study population
Age (years) (mean or median) Male (%) BCLC stage (%) Child–Pugh class (%)
Kudo 2021 [32]

NCT01658878,

CheckMate 040

1/2 Multi-centre

• Non-Randomized

• Parallel Assignment

• Open Label

67 NA

4(A), 16(B), 73(C),

NR(D)

2(A6), 76(B7), 22(B8)
Yau 2019a [33]

NCT02576509,

CheckMate 459

3 Multi-centre

• Randomized

• Parallel Assignment

• Open Label

64.2 84.9 NA NA
Finn 2020 [41] NCT03006926 1 Multi-centre

• NA

• Single Group Assignment

• Open Label

66.5 81.0 29(B), 71(C) 71(A5), 27(A6), 2(B7)
Finn 2020 [13]

NCT03434379,

IMbrave 150

3 Multi-centre

• Randomized

• Parallel Assignment

• Open Label

Atezo + Bev 64

SOR 66

Atezo + Bev 82

SOR 83

Atezo + Bev

2(A), 15(B), 82(C)

SOR

4(A), 16(B), 81(C)

Atezo + Bev

72(A5), 28(A6)

SOR

73(A5), 27(A6)

Xu 2021 [42]

NCT03463876

RESCUE

2 Mainland China

• NA

• Single Group Assignment

• Open Label

1-L 53

2-L 51

1-L 90.0

2-L 88.3

1-L

17.1(B), 82.9(C)

2-L

18.3(B), 81.7(C)

1-L

87.1(A5), 12.9(A6)

2-L

84.2(A5), 15.8(A6)

Kim 2021a [43] NCT03347292 1b United States

• Non-Randomized

• Sequential Assignment

• Open Label

67 NA 41(B), 55(C) 100(A)
Jiao 2021a [44] NCT04344158 3 Mainland China

• Randomized

• Parallel Assignment

• Open Label

56 NA 23(B), 77(C) NA
Kudo 2020a [45]

NCT03418922

Study 117

1b Japan

• Non-Randomized

• Sequential A ssignment

• Open Label

NA NA NA NA
Kudo 2020 [46]

NCT03289533

VEGF Liver 100

1 Japan

• Non-Randomized

• Parallel Assignment

• Open Label

68.5 90.9 40.9(B), 59.1(C) NA
Lee 2020 [35]

NCT02715531

GO30140

1b Multi-centre

• Randomized

• Parallel Assignment

• Open Label

A 62

F1 60

F2 63

A 81

F1 90

F2 83

A 0(A), 10(B), 90(C)

F1 0(A), 10(B), 90(C)

F2 3(A), 7(B), 90(C)

A 74(A5), 20(A6), 6(B7)

F1 72(A5), 28(A6), 0(B7)

F2 71(A5), 29(A6), 0(B7)

Li 2021 [52] NCT03092895 1b/2 Mainland China

• Non-Randomized

• Parallel Assignment

• Open Label

52 91.2 11.8(B), 85.3(C), 2.9(unknown) 97.1(A), 2.9(B)
Lin 2021a [47] ChiCTR1900028295 2 Mainland China

• NA

• Single arm

• Open Label

NA NA NA 100(≤ B7)
Ren 2021 [36]

NCT03794440

ORIENT-32

3 Mainland China

• Randomized

• Parallel Assignment

• Open Label

Sintilimab + IBI305 53

SOR 54

Sintilimab + IBI305 88

SOR 90

Sintilimab + IBI305

15(B), 85(C)

SOR

14(B), 86(C)

Sintilimab + IBI305

96(A), 4(B)

SOR

95(A), 5(B)

Kelley 2022 50]

NCT03755791

COSMIC-312

3 Multi-centre

• Randomized

• Parallel Assignment

• Open Label

Cabozantinib + Atezo 64

SOR 64

Cabozantinib + Atezo 83

SOR 86

Cabozantinib + Atezo 32(B) 68(C)

SOR 33(B) 67(C)

Cabozantinib + Atezo 100(A)

SOR 100(A)

He 2021a [53] NCT04044313 2 Mainland China

• NA

• Single Group Assignment

• Open Label

49 91.7 NA NA
Abou-Alfa 2022a [54]

NCT03298451

HIMALAYA

3 Multi-centre

• Randomized

• Parallel Assignment

• Open Label

NA NA NA NA
Bai 2021a [48] NCT04444167 2 Mainland China

• NA

• Single Group Assignment

• Open Label

52.5 86.7 NA NA
Verset 2022 [34]

NCT02702414

KEYNOTE-224

2 Multi-centre

• NA

• Single Group Assignment

• Open Label

68 86 22(B), 78(C) 100(A)
Chen 2022 [51] NCT04052152 2 Mainland China

• NA

• Single Group Assignment

• Open Label

56 90.0 25(B), 75(C) 95(A), 5(B)
Hao 2022a [37] NCT04605796 2 Mainland China

• NA

• Single Group Assignment

• Open Label

54 88.9 74.1(C) NA
Meyer 2022a [38] NCT03468426 1b Multi-centre

• NA

• Single Group Assignment

• Open Label

1-L 65

2-L 64

1-L 87

2-L 77

NA NA
Lim 2022a [39] NCT02519348 2 Multi-centre

• Randomized

• Parallel Assignment

• Open Label

NA NA NA NA
Yoo 2022a [49]

NCT04310709

RENOBATE

2 Korea

• NA

• Single Group Assignment

• Open Label

61 (40–79) 73.8 90.5(C) NA
Maesaka 2022 [40] NA NA Japan

• NA

• Parallel Assignment

• Open Label

Atezo + Bev 76

Len 73

Atezo + Bev 76.8

Len 76.3

Atezo + Bev

49.3(A/B), 50.7(C)

Len

40.7(A/B), 50.3(C)

Atezo + Bev

97.1(A), 2.9(B)

Len

79.5(A), 20.5(B)

Author, year Study drug(s), n Comparator Follow-up time (mo) Outcome(s) studied
PFS median, mo OS median, mo ORR (%) DCR (%) TRAEs (%)
Kudo 2021 [32] Nivo (SOR naïve), 25 Nivo (SOR treated), 24 16.3 (12.2–22.5)

1-L 3.4 (1.6–4.1)

2-L 2.2 (1.4–4.2)

1-L 9.8 (3.7–14.3)

2-L 7.4 (2.3–12.1)

1-L 12

2-L 13

1-L 60

2-L 50

Any grade:

1-L 44

2-L 58

Yau 2019a [33] Nivo, 371 SOR, 372 NA

Nivo 3.68 (3.06–3.88)

SOR 14.69 (11.89–17.22)

Nivo 16.39 (13.93–18.37)

SOR 14.69 (11.89–17.22)

Nivo 15.4

SOR 7.0

NA

SAEs:

Nivo 56.40

SOR 58.95

Finn 2020 [41] Len + Pembro, 100 NA 10.6 (9.2–11.5) 8.2 (7.4–9.7) 22.0 (20.4-NE) 46 86 Grade ≥ 3 TRAEs: 67
Finn 2020 [13] Atezo + Bev, 336 SOR, 165

Atezo + Bev 8.9 (7.1–11.1)

SOR 8.1 (4.7–10.2)

Atezo + Bev 6.83 (5.75–8.28)

SOR 4.27 (3.98–5.55)

Atezo + Bev NE

SOR 13.2 (10.4-NE)

Atezo + Bev 27.3

SOR 11.9

Atezo + Bev 73.6

SOR 55.3

Any grade:

Atezo + Bev 98.2

SOR 98.7

Xu 2021 [42] Cam + Apa (1L), 70 Cam + Apa (2L), 120

1-L 16.7 (11.1–18.2)

2-L 14.0 (9.6– 17.0)

1-L 5.7 (5.4 -7.4)

2-L 5.5 (3.7–5.6)

1-L NE

2-L NE

1-L 34.3

2-L 22.5

1-L 77.1

2-L 75.8

1-L Grade ≥ 3: 78.6

2-L Grade ≥ 3: 76.7

Kim 2021a [43] Reg + Pembro, 29 NA NA NA NA NA NA 24
Jiao 2021a [44] Penpulimab + Anlotinib, 31 NA 11.9 (3.7–17.7) 7.6 NE 31 82.8 Grade ≥ 3: 16.1
Kudo 2020a [45] Len + Nivo, 24 NA NA NA NA 79.2 NA NA
Kudo 2020 [46] Avelumab + axitinib, 22 NA NA 5.52 (1.91–7.39) 14.05 (7.95-NE) 13.6 68.2 Grade 3–4: 77.2
Lee 2020 [35] A: Atezo + Bev, 104

F1: Atezo + Bev, 60

F2: Bev, 59

A 6.6 (5.5–8.5)

F1 6.6 (5.5–8.5)

F2 6·7 (4.2–8.2)

A 7.3 (5.4–9.9)

F1 5.6 (3.6–7.4)

F2 3.4 (1.9–5.2)

A NE

F1 NE

F2 NE

A 36

F1 20

F2 17

A 71

F1 67

F2 49

Grade 3–4: A 53

F1 17

F2 5

Li 2021 [52] Cam + FOLFOX4, 34 NA 11.5 (2.7–22.4) 7.4 (3.9- 9.2)

6 mo 79.4%

12 mo 50.0%

29.4 79.4 Grade ≥ 3 TRAEs: 85.3
Lin 2021a [47] Anlotinib + toripalimab, 30 NA NA NA NA 25 87.5 Grade 3: 45.5
Ren 2021 [36] Sintilimab + IBI305, 380 SOR, 191

Sintilimab + IBI305 10.0 (8.5–11.7)

SOR 10.0 (8.4–11.7)

Sintilimab + IBI305 4.6 (4.1–5.7)

SOR 2.8 (2.7–3.2)

NA

Sintilimab + IBI305 21

SOR 4

Sintilimab + IBI305 4.6 72

SOR 64

Grade ≥ 3:

Sintilimab + IBI305 55

SOR 48.1

Kelley 2022 [50] Atezo + Cabozantinib, 432

SOR, 217,

Cabozantinib, 188

15.8 (14.5–17.2)

Cabozantinib + Atezo 6.8 (99% CI 5.6–8.3)

SOR 4.2 (99% CI 2.8–7.0)

Cabozantinib + Atezo 15.4 (96% CI 13.7–17.7)

SOR 12.2 (96% CI 15.5-NE)

Cabozantinib + Atezo 11

SOR 4

Cabozantinib + Atezo 78

SOR 65

Any grade: 93
He 2021a [53] Toripalimab + LEN + HAIC, 36 NA 11.2 10.5 (6.21 − 14.79) NA 63.9 NA Grade ≥ 3: 72.2
Abou-Alfa 2022a [54] Tremelimumab + durvalumab, 393

Durvalumab, 389,

SOR, 389

STRIDE 16.1

Durvalumab 16.5

SOR 13.3

STRIDE 3.8 (3.7–5.3)

Durvalumab 3.7 (3.2–3.8)

SOR 4.1 (3.8–5.5)

STRIDE 16.4 (14.2–19.6)

Durvalumab 16.6 (14.1–19.1)

SOR 13.8 (12.3–16.1)

STRIDE 20.1

D 17.0

S 5.1

NA Grade ≥ 3: 25.8
Bai 2021a [48] AK104 + LEN, 30 NA NA NA NA 44.4 77.8 Any grade: 83.3
Verset 2022 [34] Pembro, 51 NA 27 (range, 23–29) 4 (2–8) 17 (8–23) 16 57 Any grade: 55
Chen 2021a [51] Sintilimab + anlotinib, 20 NA 12 (range 3–19) 12.2(3.8-NR) NA 40 95 Any grade: 100
Hao 2022a [37] Toripalimab + Bev, 54 NA NA 9.9 (5.5–11.0) NE 32.7 78.8 Grade ≥ 3: 25.9
Meyer 2022a [38] Ezabenlimab + BI 836,880, 1-L 30 Ezabenlimab + BI 836,880, 2-L 31 NA NA NA 21 85.7 Any grade: 48
Lim 2022a [39] Durvalumab + Bev, 47 NA NA NA NE 21.3 NA Any grade: 70.2
Yoo 2022a [49] Nivo + regorafenib, 42 NA 9.2 (8.5–9.9) 5.5 (1.8–9.1) NE 31 NA NA
Maesaka 2022 [40] Atezo + Bev, 69 LEN, 161 NA

Atezo + Bev 8.8

LEN 5.2

Atezo + Bev NR

LEN 20.6

Atezo + Bev 29.7

LEN 30.2

Atezo + Bev 71.9

LEN 82.5

Any grade: 98.5

1-L, first-line; 2-L, second-line; Atezo, atezolizumab; BCLC, Barcelona Clinic Liver Cancer; Bev, bevacizumab; Cam, camrelizumab; FOLFOX4, fluorouracil, leucovorin, and oxaliplatin; LEN, lenvatinib; mo, month; NA, not available; NE, not estimable; Nivo, nivolumab; Pembro, pembrolizumab; REG, regorafenib; SOR, sorafenib; SAEs, serious adverse events; STRIDE, tremelimumab plus durvalumab; TRAEs, treatment-related adverse events

aConference abstract