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. 2022 Sep 26;13(10):1648–1654. doi: 10.1021/acsmedchemlett.2c00336

Figure 3.

Figure 3

SAR study of the warhead. FP screening of a panel of acrylamide-based molecules with an extended warhead against both zDHHC20 and zDHHC2, with activity normalized to DMSO. Compounds were screened at 10 μM. Data are presented as mean ± standard deviation (n = 3).