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Enzyme inhibition profiling of 3–9 and calpeptin.
| compound | IC50 (μM) | aKD (μM) |
|---|---|---|
| 3 | >425 | >2.13 E+02 |
| 4 | 2.51 ± 0.24 | 1.26 ± 0.12 |
| 5 | >213 | >1.07 E+02 |
| 6 | 37.84 ± 5.23 | 18.92 ± 2.61 |
| 7 | >425 | >2.13 E+02 |
| 8 | 197.73 ± 23.77 | 98.86 ± 11.89 |
| 9 | >170 | >8.50 E+01 |
| 57 | 6.49 ± 0.73 | 3.26 ± 0.36 |
| 58 | 2.37 ± 0.81 | 1.19 ± 0.40 |
| calpeptin | 2.43 ± 0.20 | 1.22 ± 0.10 |
calculated by using the Cheng Prussoff equation.
