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. 2022 Aug 2;13(10):1234–1238. doi: 10.1039/d2md00150k

Antibacterial activity of selected carborane–cyclam conjugates against Mtb strain H37Rv.

Compound MIC (μM) Ref.
1 3.13 13
9 0.80 This work
Cs2·10 0.78
14 3.22
Cs2·15 nda
19 0.64
Cs2·20 nda
Rifampicin 0.06 Controls
Isoniazid 0.16
a

nd = not determined.