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. 2022 Jul 20;13(10):1246–1264. doi: 10.1039/d2md00153e

Effects of various five-membered heteroaromatic rings on the kinase inhibitory activity of diphenylpyrimidine–diamine derivatives.

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Cpd. R3 R4 Axl IC50 (nM) Cpd. R3 R4 Axl IC50 (nM)
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