Skip to main content
. 2022 Jul 20;13(10):1246–1264. doi: 10.1039/d2md00153e

Pharmacokinetic data of compounds m6, m16, and TP-0903 in rats.

Parameter m6 m16 TP-0903
PO 5 mg kg−1 IV 1 mg kg−1 PO 5 mg kg−1 IV 1 mg kg−1 PO 5 mg kg−1 IV 1 mg kg−1
AUClast (ng h−1 mL−1) 661 497 1180 422 158 187
C max (ng mL−1) 169 337 83.9 56.3 46.8 89.8
CL (mL h−1 kg−1) NA 1.95 NA 2.20 NA 4.97
T 1/2 (h) 1.32 1.49 6.45 6.6 2.94 1.77
F% 26.6 56.1 21.5