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. 2022 Oct 4;45(5):171–175. doi: 10.18773/austprescr.2022.063

Table 2. Commonly prescribed drugs with significant CFTR-modulator interactions involving cytochrome P450 3A4.

CYP3A4 inducers CYP3A4 inhibitors
Barbiturates (phenobarbital) Azole antifungals
Carbamazepine Amiodarone
Phenytoin Erythromycin
Rifampicin Clarithromycin
St John’s wort Protease inhibitors (ritonavir)

CFTR cystic fibrosis transmembrane conductance regulator

CYP cytochrome P450