Table 2. Commonly prescribed drugs with significant CFTR-modulator interactions involving cytochrome P450 3A4.
| CYP3A4 inducers | CYP3A4 inhibitors |
|---|---|
| Barbiturates (phenobarbital) | Azole antifungals |
| Carbamazepine | Amiodarone |
| Phenytoin | Erythromycin |
| Rifampicin | Clarithromycin |
| St John’s wort | Protease inhibitors (ritonavir) |
CFTR cystic fibrosis transmembrane conductance regulator
CYP cytochrome P450