Table 3.

GP values calculated as GP = (I₄₄₀ − I₄₉₀)/(I₄₄₀ + I₄₉₀) before and after the treatment with the peptide [Nle¹, dLeu⁹, dLys¹⁰]TL. The GP values of lead peptide [dLeu⁹, dLys¹⁰]TL was calculated previously [27].

GP Value
LUVs: DOPG/CL
cmpd	Unloaded LUVs	LUVs + 5 μM cmpd	LUVs + 30 μM cmpd
[dLeu9, dLys10]TL	−0.18 ± 0.01	−0.06 ± 0.01	0.26 ± 0.02
[Nle1, dLeu9, dLys10]TL	−0.18 ± 0.01	0.03 ± 0.01	0.29 ± 0.03
LUVs: DOPG/DOPE/CL
cmpd	Unloaded LUVs	LUVs + 5 μM cmpd	LUVs + 30 μM cmpd
[dLeu9, dLys10]TL	−0.07 ± 0.01	0.09 ± 0.02	0.11 ± 0.02
[Nle1, dLeu9, dLys10]TL	−0.07 ± 0.01	0.05 ± 0.01	0.13 ± 0.03