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The eticlopride analogues 13, 15, 17b, 48, 49 were all antagonists or very weak partial agonists at both D3R and D2R. The Go BRET activation assays show that these compounds have very low efficacies at both D3R (A) and D2R (B) similar to levels of the reference antagonist eticlopride, compared to the full agonist quinpirole.
