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. 2022 Oct 17;65(20):13505–13532. doi: 10.1021/acs.jmedchem.2c01177

Table 1. Exosites in ADAMTS4 and ADAMTS5a.

enzyme region exosite ref
ADAMTS4 Sp 717QGNPGHRS724 (22)
ADAMTS4 Sp 788AGNPQDTR795 (22)
ADAMTS5 Sp 739NKKSKG744 (22)
ADAMTS5 Sp 837TDPTKPLD844 (22)
ADAMTS5 Dis 532KK533 (51)
a

Abbreviations: Dis, disintegrin-like domain; Sp, spacer domain.