Table 1.
Antimicrobial and Hemolytic Activities of Peptoids
| MIC [μg mL−1]a |
||||||
|---|---|---|---|---|---|---|
| peptoid/sequence | chemical formula | S. aureus | P. aeruginosa | A. baumannii | HC50 [μg mL−1]b | SRc |
| L1/Ac(NapNdp)3 | C65H86N10O7 | 15.6 | 15.6 | 15.6 | >250 | >16 |
| C1/C(NapNdp)3 | C63H81N9O6 | 3.9 | 7.8 | 7.8 | >250 | >64 |
| L2/Ac(NapNnm)3 | C56H68N10O7 | 125 | 125 | 125 | >250 | >2 |
| C2/C(NapNnm)3 | C54H63N9O6 | 31.3 | 31.3 | 31.3 | >250 | >8 |
Minimum inhibitory concentrations against Staphylococcus aureus, Pseudomonas aeruginosa, and Acinetobacter baumannii.
Hemolytic concentrations at which 50% hemolysis is observed.
Selectivity ratio: HC50/MIC against S. aureus.