Table 2. Species Cross Reactivity and Selectivity Binding Data for Fluorescein-Labeled Bicycle 2 As Determined by FP Direct Binding.
species cross reactivity | selectivity | |||||
---|---|---|---|---|---|---|
protein | human Nectin-4 ECD | mouse Nectin-4 ECD | rat Nectin-4 ECD | NHP (Cyno) Nectin-4 ECD | Nectin 1–3, 5 ECD | Nectin-like 1–5 ECD |
Kd (nM) | 19.4 | 42.9 | 91.8 | 49.2 | >2000 | >2000 |