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. 2022 Oct 7;65(21):14337–14347. doi: 10.1021/acs.jmedchem.2c00065

Table 2. Species Cross Reactivity and Selectivity Binding Data for Fluorescein-Labeled Bicycle 2 As Determined by FP Direct Binding.

  species cross reactivity selectivity
protein human Nectin-4 ECD mouse Nectin-4 ECD rat Nectin-4 ECD NHP (Cyno) Nectin-4 ECD Nectin 1–3, 5 ECD Nectin-like 1–5 ECD
Kd (nM) 19.4 42.9 91.8 49.2 >2000 >2000