Table 4. Affinities of Compound 10 Analogues Containing Non-Natural Amino Acids Determined by FP Competition^a.

^aAffinities were measured using fluorescence polarization competition. The Geomean of K_i values displayed are all generated from n ≥ 2. Full assay details, including the number of replicates, errors, and competing tracer molecule are in the Supporting Information. Amino acid sequence of parent peptide 10 Ac-CPFGCMKNWSWPIWC–CONH₂ (TATA scaffold).