Table 5. BCAT1 and BCAT2 Activities of Annulated Compounds and Intestinal Caco-2 Permeabilitiesa.
IC50 values given are arithmetic mean values over at least two independent IC50 determinations.
Compounds 35, 36, and 37 are racemates.
IC50 values given are arithmetic mean values over at least two independent IC50 determinations.
Compounds 35, 36, and 37 are racemates.