Table 2. Selectivity Profiles of 30 in Binding and Cellular Assays.
| assay | IC50 (nM) |
|---|---|
| JAK1 JH1 | >1000 |
| JAK2 JH1 | >1000 |
| JAK3 JH1 | >1000 |
| TYK2 JH1 | >1000 |
| EPO | 3496 |
| IL-2 | 41 |
| IL-6 | 33 |
| assay | IC50 (nM) |
|---|---|
| JAK1 JH1 | >1000 |
| JAK2 JH1 | >1000 |
| JAK3 JH1 | >1000 |
| TYK2 JH1 | >1000 |
| EPO | 3496 |
| IL-2 | 41 |
| IL-6 | 33 |