Table 2. Selectivity Profiles of 30 in Binding and Cellular Assays.
assay | IC50 (nM) |
---|---|
JAK1 JH1 | >1000 |
JAK2 JH1 | >1000 |
JAK3 JH1 | >1000 |
TYK2 JH1 | >1000 |
EPO | 3496 |
IL-2 | 41 |
IL-6 | 33 |
assay | IC50 (nM) |
---|---|
JAK1 JH1 | >1000 |
JAK2 JH1 | >1000 |
JAK3 JH1 | >1000 |
TYK2 JH1 | >1000 |
EPO | 3496 |
IL-2 | 41 |
IL-6 | 33 |