Skip to main content
. Author manuscript; available in PMC: 2022 Nov 21.
Published in final edited form as: J Med Chem. 2020 Jan 24;63(3):1298–1312. doi: 10.1021/acs.jmedchem.9b01769

Table 9.

Inhibition of hERG potassium channel activity by 24b in HEK293 cells.

cell hERG inhibitory effect (%)
0.3 μM 1 μM 3 μM 10 μM 30 μM
cell 1 4.12 8.01 13.35 18.48 21.59
cell 2 1.75 NA NA NA NA
cell 3 NA 9.21 11.90 18.96 22.85
Mean (%) 2.93 8.61 12.63 18.72 22.22
SD 1.68 0.84 1.03 0.33 0.89