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. 2022 Nov 28;12(52):34126–34141. doi: 10.1039/d2ra03226k
GI50 values (M) mean ± SD Selectivity indices (SI)
MCF-7 HCT-116 MRC-5 MCF-7 HCT-116 MW c log Pc LE (MCF-7) LE (HCT-116) tPSAd Nrotd HBAd HBDd
graphic file with name d2ra03226k-u34.jpg
l 9.2 ± 0.4 8.4 ± 0.9 30.1 ± 0.6 3.3 3.6 364.4 3.75 0.26 0.27 108 6 6 1
m 2.0 ± 0.8 4.7 ± 1.3 16.5 ± 0.6 8.3 3.5 440.4 5.43 0.26 0.24 89 6 4 1
n 25.4 ± 1.6 1.1 ± 0.5 12.1 ± 0.4 0.5 11 373.3 4.97 0.26 0.34 89 4 4 1