GI50 values (M) mean ± SD | Selectivity indices (SI) | ||||||||||||
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
MCF-7 | HCT-116 | MRC-5 | MCF-7 | HCT-116 | MW | c log Pc | LE (MCF-7) | LE (HCT-116) | tPSAd | Nrotd | HBAd | HBDd | |
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s | 7.3 ± 0.8 | 8.4 ± 0.6 | 18.1 ± 0.4 | 2.5 | 2.2 | 364.4 | 3.43 | 0.27 | 0.27 | 119 | 6 | 6 | 2 |
t | 4.5 ± 1.4 | 6.5 ± 2.6 | 13.2 ± 0.3 | 2.9 | 2 | 332.4 | 4.54 | 0.30 | 0.29 | 89 | 4 | 4 | 1 |
u | 12.8 ± 0.7 | 27.2 ± 0.5 | 30.4 ± 0.2 | 2.4 | 1.1 | 373.3 | 5 | 0.28 | 0.26 | 89 | 4 | 4 | 1 |