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. 2022 Nov 28;12(52):34126–34141. doi: 10.1039/d2ra03226k
GI50 values (M) mean ± SD Selectivity indices (SI)
MCF-7 HCT-116 MRC-5 MCF-7 HCT-116 MW c log Pc LE (MCF-7) LE (HCT-116) tPSAd Nrotd HBAd HBDd
graphic file with name d2ra03226k-u36.jpg
s 7.3 ± 0.8 8.4 ± 0.6 18.1 ± 0.4 2.5 2.2 364.4 3.43 0.27 0.27 119 6 6 2
t 4.5 ± 1.4 6.5 ± 2.6 13.2 ± 0.3 2.9 2 332.4 4.54 0.30 0.29 89 4 4 1
u 12.8 ± 0.7 27.2 ± 0.5 30.4 ± 0.2 2.4 1.1 373.3 5 0.28 0.26 89 4 4 1