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. 2022 Nov 15;82(16):1621–1627. doi: 10.1007/s40265-022-01800-5

Key clinical trials of valemetostat

Drug(s) Indication Phase Status Location(s) Sponsor/Collaborator Identifier
Valemetostat R/R ATL 2 Ongoing Japan Daiichi Sankyo NCT04102150; JapicCTI-194964
Valemetostat R/R PTCL 2 Ongoing Global Daiichi Sankyo NCT04703192; EudraCT2020-004954-31; jRCT2071200095; VALENTINE-PTCL01
Valemetostat R/R NHL (including BCL, ATL and PTCL) 1 Ongoing Japan, USA Daiichi Sankyo NCT02732275; JapicCTI-163173
Valemetostat R/R BCL 2 Ongoing Belgium, France The Lymphoma Academic Research Organisation; Daiichi Sankyo NCT04842877; EudraCT2020-005225-81; VALYM
Valemetostat AML or ALL 1 Terminateda USA Daiichi Sankyo NCT03110354
Valemetostat, irinotecan Recurrent SCLC 1/2 Ongoing USA Memorial Sloan Kettering Cancer Center NCT03879798
Valemetostat, ipilimumab Metastatic prostate, urothelial, and renal cell cancers 1 Ongoing USA M.D. Anderson Cancer Center; National Cancer Institute NCT04388852; NCI-2020-02916
Valemetostat Malignant solid tumoursb 1 Ongoing Japan National Cancer Center Hospital, Tokyo

jRCT2031190268

NCCH1904/MK007; ELEPHANT

AML acute myelogenous leukaemia, ALL acute lymphocytic leukaemia, ATL adult T-cell leukaemia/lymphoma, BCL B-cell lymphoma, NHL non-Hodgkin lymphoma, PTCL peripheral T-cell lymphoma, R/R relapsed/refractory, SCLC small cell lung cancer

aTerminated because of slow patient accrual

bIn children, adolescents and young adults aged 3–29 years