TABLE 2.
Inhibition profile of P. gingivalis DPPIV
| Inhibitor | Concn | % of residual activity |
|---|---|---|
| DFP | 1 mM | 0 |
| PMSF | 10 mM | 20 |
| Pefabloc | 1 mg/ml | 3 |
| 3,4-Dichloroisocoumarin | 1 mM | 100 |
| Iodoacetamide | 0.1 mM | 110 |
| N-ethylmaleimide | 5 mM | 100 |
| 1,10-Orthophenanthroline | 1 mM | 97 |
| EDTA | 10 mM | 100 |
| Leupeptin | 0.1 mM | 100 |
| Antipain | 0.1 mM | 100 |
| Prolinal | 0.1 mM | 20 |
| Cysteine | 10 mM | 105 |
| Gly-Pro | 10 mM | 200 |
| Ala-Pro | 10 mM | 30 |
| Val-Pro | 10 mM | 0 |
| Ala-Pro-Gly | 10 mM | 0 |
| Zn2+ | 1 mM | 1 |
| Hg2+ | 1 mM | 3 |
| SDS | 1% | 0 |
| Triton X-100 | 1% | 0 |