TABLE 2.
Inhibition profile of P. gingivalis DPPIV
Inhibitor | Concn | % of residual activity |
---|---|---|
DFP | 1 mM | 0 |
PMSF | 10 mM | 20 |
Pefabloc | 1 mg/ml | 3 |
3,4-Dichloroisocoumarin | 1 mM | 100 |
Iodoacetamide | 0.1 mM | 110 |
N-ethylmaleimide | 5 mM | 100 |
1,10-Orthophenanthroline | 1 mM | 97 |
EDTA | 10 mM | 100 |
Leupeptin | 0.1 mM | 100 |
Antipain | 0.1 mM | 100 |
Prolinal | 0.1 mM | 20 |
Cysteine | 10 mM | 105 |
Gly-Pro | 10 mM | 200 |
Ala-Pro | 10 mM | 30 |
Val-Pro | 10 mM | 0 |
Ala-Pro-Gly | 10 mM | 0 |
Zn2+ | 1 mM | 1 |
Hg2+ | 1 mM | 3 |
SDS | 1% | 0 |
Triton X-100 | 1% | 0 |