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. 2022 Nov 29;9:1067516. doi: 10.3389/fmed.2022.1067516

TABLE 3.

MICs of the four novel oxazolidinones for the Mtb clinical isolates with different MICs of linezolid.

Linezolid No. of isolates with different MICs (μg/ml)


MIC (μg/ml) No. of isolates Contezolid Tedizolid Sutezolid Delpazolid
≤ 0.0625 3 ≤ 0.0625 (2)
0.25 (1)
≤ 0.0625 (3) ≤ 0.0625 (3) ≤ 0.0625 (1)
0.25 (1)
1 (1)
0.125 10 ≤ 0.0625 (3)
0.125 (2)
0.25 (4)
0.5 (1)
≤ 0.0625 (8)
0.125 (1)
0.5 (1)
≤ 0.0625 (10) 0.25 (5)
0.5 (4)
1 (1)
0.25 28 ≤ 0.0625 (6)
0.125 (1)
0.25 (4)
0.5 (17)
≤ 0.0625 (11)
0.125 (6)
0.25 (8)
0.5 (2)
1 (1)
≤ 0.0625 (26)
0.125 (2)
0.25 (2)
0.5 (8)
1 (16)
2 (2)
0.5 26 0.125 (1)
0.5 (22)
1 (3)
0.125 (11)
0.25 (12)
0.5 (3)
≤ 0.0625 (25)
0.25 (1)
0.5 (4)
1 (7)
2 (14)
4 (1)
1 2 0.5 (2) 0.125 (2) ≤ 0.0625 (2) 1 (2)