Table 1.
Drugs Included in the Screen
Drug | Target/Mechanism of Action | Clinical Trials Phase | References |
---|---|---|---|
Trabectedin | RNA Pol II, DNA-bound proteins, tumor microenvironment/multitarget DNA-damaging agent | III | Monk et al.36 |
CX-4945 | Casein kinase 2, Cdc2-like kinases | Ib/II | Borad et al.37 |
Foretinib | C-MET, VEGFR2, TAM (TYRO, Axl, MERTK) receptors | II | Rayson et al.38 |
RG7112 | MDM2–p53 interaction/p53 activator | I | Andreeff et al.39 |