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. 2022 Oct 31;10(6):e02592-22. doi: 10.1128/spectrum.02592-22

TABLE 4.

Interacting residues of HadAB with NSC19723 and thiacetazone

Compound Chain Binding site residues type
Acidic Basic Polar Hydrophobic
NSC19723 HadA G64, Y65, Q68, Q86, Q89, N125, T138, T140 I60, C61, V62, L91, C105, V127,
HadB D36 Y30, S34 M60
Thiacetazone HadA Y28, G64, Y65, Q68, Q86, N125, T138, T140 C61, V62,
HadB D36 H58 Y30, S34 M60