Table 12.
Serum Effects on MRSA MIC of Lead 4-Aminoquinoline and 5-Amino-4-quinolone Compounds
compd | MIC (μg/mL) | MIC + 10% FBS (μg/mL) | MIC + 10% mouse serum (μg/mL) |
---|---|---|---|
22 | 0.0625 | 8 | |
31 | 0.25 | 4–8 | |
111 | <0.0625 | 4 | 4–8 |
120 | 0.125 | 4 |
Serum Effects on MRSA MIC of Lead 4-Aminoquinoline and 5-Amino-4-quinolone Compounds
compd | MIC (μg/mL) | MIC + 10% FBS (μg/mL) | MIC + 10% mouse serum (μg/mL) |
---|---|---|---|
22 | 0.0625 | 8 | |
31 | 0.25 | 4–8 | |
111 | <0.0625 | 4 | 4–8 |
120 | 0.125 | 4 |