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. Author manuscript; available in PMC: 2024 Jan 1.
Published in final edited form as: Biomed Pharmacother. 2022 Nov 29;157:114047. doi: 10.1016/j.biopha.2022.114047

Table 3:

ADCs cytotoxicity on human tumor cells.

IC50 (nM) MDA-MD-468 BT20 A431 MDA-MB-231
40H3-Tesirine 0.3097 9.066 1.847 >100
40H3-MCVCPAB-MMAE 3.446 18.58 9.125 >100
40H3-CL2A-SN38 27.83 98.812 19.71 >100
40H3-SMCC-DM1 6.652 >100 89.6 >100
40H3-Deruxtecan 9.316 70.361 90.21 >100
40H3 > 100 >100 >100 >100