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. 2023 Jan 11;38(1):2152810. doi: 10.1080/14756366.2022.2152810

Table 3.

In-vitro PIM-1 and PIM-2 kinase inhibition data of the most active compounds.

Code PIM-1
IC50 (µM)
PIM-2
IC50 (µM)
5b 1.31 0.67
5c 1 1.66
6e 1.10 1.49
13a 1.27
13c 7.78
14a 0.385
Quercetin 1.17 0.61