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. 2022 Dec 28;16(1):43. doi: 10.3390/ph16010043

Table 3.

% Inhibition values of the synthesized lapatinib derivatives 6al over EGFR and HER2 kinases at 10 µM.

Cpd % Kinase Inhibition at 10 µM
EGFR HER2
6a 98.79 74.72
6b 99.34 78.04
6c 99.32 89.99
6d 99.09 79.68
6e 67.27 8.78
6f 76.55 11.69
6g 91.80 43.06
6h 94.67 47.34
6i 97.65 87.16
6j 99.03 96.73
6k 98.64 91.16
6l 98.58 89.05