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. Author manuscript; available in PMC: 2024 Feb 1.
Published in final edited form as: Curr Opin Chem Biol. 2022 Dec 28;72:102255. doi: 10.1016/j.cbpa.2022.102255

Figure 1. Small molecule KAT inhibitors.

Figure 1.

Representative small molecule inhibitors of p300/CBP (top) and MYST (bottom) family acetyltransferases that have been linked to pharmacological studies described here. All the depicted p300/CBP inhibitors are active site competitive, except where parenthetically noted. MYST family member isoform selectivity is noted parenthetically.